GSK2879552 free base CAS 1401966-69
GSK2879552 is an orally available, irreversible inhibitor of lysine specific demethylase 1 (LSD1; officially known as lysine demethylase 1A, KDM1A). It was investigated for potential to modulate epigenetic regulation in cancer, but the programme was terminated due to serious adverse events becoming evident in early trials
Technical Data for GSK2879552
| M. Wt | 364.48 |
| Formula | C23H28N2O2 |
| Storage | Store at +4°C |
| Purity | ≥99% (HPLC) |
| CAS Number | 1401966-69-5 |
| Appearance | Solid |
| InChI Key | LRULVYSBRWUVGR-FCHUYYIVSA-N |
| Smiles | C1CN(CCC1CNC2CC2C3=CC=CC=C3)CC4=CC=C(C=C4)C(=O)O |
Synonyms
GSK2879552
1401966-69-5
GSK-2879552
UNII-GT77Z6Y09Z
4-((4-((((1R,2S)-2-Phenylcyclopropyl)amino)methyl)piperidin-1-yl)methyl)benzoic acid